SCHEMBL4774004

SCHEMBL4774004

COc1ccc(-c2cc(-c3cc(Cl)cc(OC)c3)c(C)n2-c2ccc(OC)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.44
CHRNA7 P36544 2/20 0.42
NPSR1 Q6W5P4 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ABL1 P00519 1/20 0.41
ABCB1 P08183 1/20 0.41
BCR P11274 1/20 0.41
PTGS2 P35354 3/20 0.40
PTGS1 P23219 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778866 0.80 CHRNA7 (0.42) GLACHRNA7NPSR1MEN1ALDH1A1
SCHEMBL4777615 0.75 CHRNA7 (0.42) CHRNA7NPSR1MEN1ALDH1A1LMNA
SCHEMBL19798359 0.72 CHRNA7 (0.67) GLACHRNA7MEN1ALDH1A1LMNA
SCHEMBL6287216 0.71 HTT (0.50) CHRNA7MEN1ALDH1A1LMNAHTT
SCHEMBL19808409 0.69 CHRNA7 (0.74) CHRNA7TP53
SCHEMBL15694897 0.68 HPGD (0.52) GLACHRNA7NPSR1MEN1ALDH1A1
SCHEMBL17052682 0.68 HPGD (0.52) GLACHRNA7NPSR1MEN1ALDH1A1
SCHEMBL4778476 0.67 TP53 (0.43) GLACHRNA7NPSR1MEN1ALDH1A1
SCHEMBL4776177 0.65 CACNA2D1 (0.45) CHRNA7PTGS2PTGS1CYP1A2CYP3A4
SCHEMBL12980511 0.65 HPGD (0.52) CHRNA7NPSR1ALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1889617-A1 Triphenyl modified 5-membered heterocycles and their use as anticancer and antiflammatory agents Freie Universität Berlin (DE) 2008-02-20 EP claimed
EP-1889617-A1 Triphenyl modified 5-membered heterocycles and their use as anticancer and antiflammatory agents Freie Universität Berlin (DE) 2008-02-20 EP disclosed