SCHEMBL4774036

SCHEMBL4774036

Cc1cccc(CNc2ncnc3[nH]c(-c4ccc(N5CCCC5)cc4C)cc23)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.50
CLK4 Q9HAZ1 7/20 0.45
EGFR P00533 5/20 0.44
AURKA O14965 1/20 0.44
RPS6KB1 P23443 1/20 0.44
CSF1R P07333 2/20 0.43
CYP3A4 P08684 4/20 0.43
TSHR P16473 4/20 0.43
ALDH1A1 P00352 4/20 0.43
HPGD P15428 4/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2C19 P33261 3/20 0.43
MAPK1 P28482 2/20 0.43
ALOX15 P16050 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CYP2C9 P11712 3/20 0.42
KDM4E B2RXH2 3/20 0.42
HSD17B10 Q99714 3/20 0.42
TP53 P04637 2/20 0.42
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4770740 0.79 EGFR (0.57) CYP1A2CLK4EGFRCSF1R
SCHEMBL4763918 0.78 EGFR (0.56) CYP1A2CLK4EGFRCSF1R
SCHEMBL7494319 0.75 EGFR (0.62) CYP1A2CLK4EGFRAURKARPS6KB1
SCHEMBL4769581 0.73 EGFR (0.63) CYP1A2CLK4EGFRCSF1R
SCHEMBL4766798 0.73 EGFR (0.59) CYP1A2CLK4EGFRAURKARPS6KB1
SCHEMBL4767245 0.73 CSF1R (0.66) CYP1A2CLK4EGFRCSF1R
SCHEMBL39893 0.72 CYP1A2 (0.58) CYP1A2CLK4CYP3A4TSHRALDH1A1
SCHEMBL4766838 0.72 CSF1R (0.60) CYP1A2CLK4EGFRCSF1RCYP3A4
SCHEMBL4766521 0.70 CSF1R (0.58) CYP1A2CLK4EGFRCSF1RCYP3A4
SCHEMBL14075269 0.68 EGFR (0.78) EGFRCSF1RALDH1A1HSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1416935-B1 4-AMINO-6-PHENYL-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES NOVARTIS AG (CH) 2008-03-12 EP claimed