SCHEMBL4774971

SCHEMBL4774971

Cc1ccc(-c2nc(N)nc3ccc(Cl)nc23)c(C)c1C

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.36
MAPK1 P28482 1/20 0.36
ADORA2A P29274 2/20 0.36
HSP90AB1 P08238 1/20 0.36
DHFR P00374 6/20 0.31
NUDT1 P36639 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4097023 0.87 ADORA2A (0.44) MAPTMAPK1ADORA2AHSP90AB1DHFR
SCHEMBL4107761 0.82 HSP90AB1 (0.44) MAPTKDM4EADORA2AHSP90AB1DHFR
SCHEMBL4106705 0.82 HSP90AB1 (0.44) MAPTKDM4EADORA2AHSP90AB1DHFR
SCHEMBL4106568 0.81 ADORA2A (0.57) MAPTMAPK1ADORA2AHSP90AB1DHFR
SCHEMBL4102481 0.81 HSP90AB1 (0.40) MAPTADORA2AHSP90AB1DHFR
SCHEMBL4109781 0.78 ADORA2A (0.42) MAPTADORA2AHSP90AB1DHFRNUDT1
SCHEMBL4108093 0.77 HSP90AB1 (0.45) MAPTMAPK1ADORA2AHSP90AB1DHFR
SCHEMBL4112502 0.75 HSP90AB1 (0.43) MAPTADORA2AHSP90AB1DHFR
SCHEMBL4102985 0.75 HSP90AB1 (0.58) MAPTKDM4EMAPK1ADORA2AHSP90AB1
SCHEMBL4103265 0.74 HSP90AB1 (0.47) ADORA2AHSP90AB1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009076-A2 SUBSTITUTED PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed