SCHEMBL4774987

SCHEMBL4774987

CN1CCN(CCNc2cc(-c3cccnc3)nc(-c3ccccn3)n2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.46
ADORA1 P30542 3/20 0.46
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
KDM5B Q9UGL1 4/20 0.45
KDM6B O15054 4/20 0.45
KDM2B Q8NHM5 3/20 0.45
KDM4C Q9H3R0 3/20 0.45
PHF8 Q9UPP1 3/20 0.45
KDM6A O15550 3/20 0.45
KDM5C P41229 3/20 0.45
CHRNA1 P02708 2/20 0.45
MAOB P27338 2/20 0.45
OPRM1 P35372 2/20 0.45
OPRK1 P41145 2/20 0.45
PDE4B Q07343 2/20 0.45
SCN5A Q14524 2/20 0.45
KDM4A O75164 2/20 0.45
KDM4B O94953 2/20 0.45
KDM3A Q9Y4C1 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769045 0.92 HDAC1 (0.48) CYP3A4CYP2C9KDM5BKDM6BKDM2B
SCHEMBL2238203 0.84 HDAC1 (0.42) CYP3A4CYP2C9KDM5BKDM6BKDM2B
SCHEMBL2238217 0.84 HDAC1 (0.42) CYP3A4CYP2C9KDM5BKDM6BKDM2B
SCHEMBL4774925 0.84 HDAC1 (0.40) CYP3A4CYP2C9KDM5BKDM6BKDM2B
SCHEMBL2240387 0.84 HDAC1 (0.42) CYP3A4CYP2C9KDM5BKDM6BKDM2B
SCHEMBL4777383 0.83 METAP1 (0.47) CYP3A4CYP2C9HIF1AROS1ALK
SCHEMBL11968349 0.79 CYP3A4 (0.47) CYP3A4CYP2C9KDM5BKDM6BKDM2B
SCHEMBL2240174 0.79 CYP3A4 (0.42) CYP3A4CYP2C9KDM5BKDM6BKDM2B
SCHEMBL2238098 0.79 PTGDR (0.53) CYP3A4CYP2C9KDM4EHIF1ACYP2A6
SCHEMBL2240945 0.79 GBA1 (0.54) CYP3A4CYP2C9HIF1ACYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed