SCHEMBL4775879

SCHEMBL4775879

O=C(CCNc1cc(-c2cccnc2)nc(-c2ccccn2)n1)N1CCNCC1S(=O)(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM6A O15550 5/20 0.44
KDM6B O15054 4/20 0.44
KDM5B Q9UGL1 4/20 0.44
KDM2B Q8NHM5 4/20 0.44
KDM4C Q9H3R0 3/20 0.44
PHF8 Q9UPP1 3/20 0.44
KDM5C P41229 3/20 0.44
KDM5A P29375 3/20 0.44
CHRNA1 P02708 2/20 0.44
MAOB P27338 2/20 0.44
OPRM1 P35372 2/20 0.44
OPRK1 P41145 2/20 0.44
PDE4B Q07343 2/20 0.44
SCN5A Q14524 2/20 0.44
KDM4A O75164 2/20 0.44
KDM4B O94953 2/20 0.44
KDM3A Q9Y4C1 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAOA P21397 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2235626 0.82 HDAC1 (0.48) KDM6AKDM6BKDM5BKDM2BKDM4C
SCHEMBL4775872 0.80 KDM6A (0.47) KDM6AKDM6BKDM5BKDM2BKDM4C
SCHEMBL2239980 0.75 CYP3A4 (0.43) KDM6AKDM6BKDM5BKDM2BKDM4C
SCHEMBL2239971 0.75 SMN1; SMN2 (0.53) KDM6AKDM6BKDM5BKDM2BKDM4C
SCHEMBL4777383 0.73 METAP1 (0.47) HDAC1HDAC6
SCHEMBL4773130 0.73 HDAC1 (0.45) KDM6AKDM6BKDM5BKDM2BKDM4C
SCHEMBL4773053 0.71 MTOR (0.44) KDM6AKDM6BKDM5BKDM2BKDM4C
SCHEMBL4774925 0.71 HDAC1 (0.40) KDM6AKDM6BKDM5BKDM2BKDM4C
SCHEMBL4769045 0.70 HDAC1 (0.48) KDM6AKDM6BKDM5BKDM2BKDM4C
SCHEMBL4773622 0.69 CYP2A6 (0.46) KDM6AKDM6BKDM5BKDM2BKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed