SCHEMBL4777508

SCHEMBL4777508

C[C@@H](Oc1c(-n2cnc3ccccc32)csc1C(=O)O)c1ccccc1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 19/20 0.50
PLK3 Q9H4B4 10/20 0.49
CYP3A4 P08684 3/20 0.47
CYP2C9 P11712 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3637492 0.76 PLK1 (0.74) PLK1PLK3CYP3A4CYP2C9
SCHEMBL4146430 0.74 PLK1 (0.50) PLK1PLK3CYP3A4CYP2C9
SCHEMBL6241399 0.73 PLK1 (0.55) PLK1PLK3
SCHEMBL2986893 0.72 PLK1 (0.73) PLK1PLK3CYP3A4CYP2C9
SCHEMBL2982011 0.72 PLK1 (0.51) PLK1PLK3CYP3A4CYP2C9
SCHEMBL2990382 0.71 PLK1 (0.72) PLK1PLK3CYP3A4CYP2C9
SCHEMBL4846733 0.71 PLK1 (0.72) PLK1PLK3CYP3A4CYP2C9
SCHEMBL3574663 0.71 PLK1 (0.72) PLK1PLK3CYP3A4CYP2C9
SCHEMBL4777503 0.71 PLK1 (0.49) PLK1PLK3CYP3A4CYP2C9
SCHEMBL4631593 0.71 PLK1 (0.87) PLK1PLK3CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924572-A1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SmithKline Beecham Corporation (US) 2008-05-28 EP disclosed
WO-2007030366-A1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed