SCHEMBL4777549

SCHEMBL4777549

CC1(COc2ccc(N3CCN(C(C=O)N4CCNCC4)CC3)cc2)Cn2cc([N+](=O)[O-])nc2O1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.58
SLC6A2 P23975 1/20 0.58
SLC6A4 P31645 1/20 0.58
KCNH2 Q12809 5/20 0.57
CACNA1C Q13936 1/20 0.36
SCN5A Q14524 1/20 0.36
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
ADRB1 P08588 1/20 0.33
SIRT6 Q8N6T7 1/20 0.33
TDP1 Q9NUW8 1/20 0.31
HTR6 P50406 1/20 0.31
ENPP2 Q13822 2/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP13 P45452 1/20 0.30
ADAM17 P78536 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14562855 0.90 KCNH2 (0.68) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
SCHEMBL3466816 0.90 KCNH2 (0.68) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
Hydrochloric Acid SCHEMBL5539596 0.89 KCNH2 (0.67) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
Hydrochloric Acid SCHEMBL5539600 0.89 KCNH2 (0.67) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
SCHEMBL5547591 0.83 KCNH2 (0.68) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
SCHEMBL5542718 0.83 KCNH2 (0.68) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
SCHEMBL5546516 0.83 KCNH2 (0.68) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
SCHEMBL3466039 0.82 PTGS1 (0.58) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
SCHEMBL2094108 0.81 KCNH2 (0.68) PTGS1SLC6A2SLC6A4KCNH2CACNA1C
SCHEMBL5542442 0.81 KCNH2 (0.68) PTGS1SLC6A2SLC6A4KCNH2CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008008480-A2 NITROHETEROARYL-CONTAINING RIFAMYCIN DERIVATIVES CUMBRE PHARMACEUTICALS INC. (US) 2008-01-17 WO disclosed