SCHEMBL4777576

SCHEMBL4777576

Cc1noc(-c2ccc(N3CCC(C(=O)N4CCN(C5CCC5)CC4)C3)cc2)n1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 10/20 0.42
ALDH1A1 P00352 3/20 0.42
GPR119 Q8TDV5 1/20 0.41
IKBKE Q14164 1/20 0.40
TBK1 Q9UHD2 1/20 0.40
TP53 P04637 2/20 0.40
ACACB O00763 1/20 0.40
ACACA Q13085 1/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4668265 1.00 HRH3 (0.42) HRH3ALDH1A1GPR119IKBKETBK1
SCHEMBL4668344 1.00 HRH3 (0.42) HRH3ALDH1A1GPR119IKBKETBK1
SCHEMBL4668242 0.97 HRH3 (0.41) HRH3ALDH1A1GPR119IKBKETBK1
SCHEMBL4666773 0.97 HRH3 (0.41) HRH3ALDH1A1GPR119IKBKETBK1
SCHEMBL4666695 0.97 HRH3 (0.41) HRH3ALDH1A1GPR119IKBKETBK1
Hydrochloric Acid SCHEMBL4668308 0.96 HRH3 (0.40) HRH3ALDH1A1GPR119IKBKETBK1
Hydrochloric Acid SCHEMBL4666655 0.96 HRH3 (0.40) HRH3ALDH1A1GPR119IKBKETBK1
SCHEMBL4667354 0.89 HRH3 (0.44) HRH3ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL4667218 0.88 HRH3 (0.44) HRH3ALDH1A1MEN1KMT2A
SCHEMBL4667342 0.86 ACKR3 (0.43) HRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802307-B1 PYRROLIDINE DERIVATIVES AS HISTAMINE RECEPTORS LIGANDS GLAXO GROUP LTD (GB) 2008-02-27 EP claimed