SCHEMBL4779609

SCHEMBL4779609

C=CCn1c(Cl)nc2c1c(=O)n(CCCCS(=O)(=O)O)c(=O)n2CCC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43
ADORA2B P29275 5/20 0.41
ADORA2A P29274 4/20 0.41
PDE4A P27815 5/20 0.40
PDE4B Q07343 5/20 0.40
PDE4C Q08493 5/20 0.40
PDE4D Q08499 5/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39
BLM P54132 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RCE1 Q9Y256 1/20 0.39
PDE5A O76074 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL836600 0.85 CYP1A2 (0.47) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL13247924 0.85 CYP1A2 (0.58) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL3115778 0.82 CYP1A2 (0.52) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL835124 0.82 CYP1A2 (0.42) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL836842 0.81 CYP1A2 (0.53) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL16076197 0.81 CYP1A2 (0.55) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL836990 0.79 CYP1A2 (0.46) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL6112635 0.79 CYP1A2 (0.44) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL3108479 0.79 CYP1A2 (0.51) CYP1A2CYP2C19RECQLADORA2BADORA2A
SCHEMBL16027932 0.79 CYP1A2 (0.44) CYP1A2CYP2C19RECQLADORA2BADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912992-A1 XANTHINE DERIVATIVES AS SELECTIVE HM74A AGONISTS SmithKline Beecham Corporation (US) 2008-04-23 EP disclosed
WO-2007017262-A1 XANTHINE DERIVATIVES AS SELECTIVE HM74A AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed