SCHEMBL4780285

SCHEMBL4780285

O=C(NC(c1cccc(F)c1)C1CC1)c1c(CN2CCOCC2)c(-c2ccccc2)nc2ccccc12

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 17/20 0.69
CYP2C9 P11712 2/20 0.69
TACR2 P21452 4/20 0.64
TRPV4 Q9HBA0 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4667527 0.93 TACR3 (0.72) TACR3CYP2C9TACR2TRPV4
SCHEMBL4665928 0.92 TACR3 (0.71) TACR3CYP2C9TACR2TRPV4
SCHEMBL8267598 0.85 TACR3 (0.78) TACR3CYP2C9
SCHEMBL4887319 0.84 TACR3 (0.67) TACR3CYP2C9TACR2TRPV4
SCHEMBL4887323 0.84 TACR3 (0.67) TACR3CYP2C9TACR2TRPV4
SCHEMBL4668623 0.84 TACR3 (0.67) TACR3CYP2C9TACR2
SCHEMBL4989018 0.83 TACR3 (0.75) TACR3CYP2C9
SCHEMBL4989012 0.83 TACR3 (0.75) TACR3CYP2C9
SCHEMBL1580871 0.83 CYP2C9 (0.76) TACR3CYP2C9
SCHEMBL4898683 0.82 TACR3 (0.68) TACR3CYP2C9TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940795-A1 N-OXO-HETEROCYCLE AND N-OXO-ALKYL QUINOLINE-4-CARBOXAMIDES AS NK-3 RECEPTOR LIGANDS AstraZeneca AB (SE) 2008-07-09 EP claimed
WO-2007035156-A1 N-OXO-HETEROCYCLE AND N-OXO-ALKYL QUINOLINE-4-CARBOXAMIDES AS NK-3 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2007-03-29 WO claimed