SCHEMBL4781934

SCHEMBL4781934

Cc1c[nH]c2ncnc(N3CCC(N)(CN(CCN(C)C)Cc4ccccc4)C3)c12

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 13/20 0.58
LIMK1 P53667 6/20 0.46
ROCK2 O75116 5/20 0.46
PRKACA P17612 5/20 0.46
PRKACG P22612 5/20 0.46
PRKACB P22694 5/20 0.46
LIMK2 P53671 4/20 0.44
ROCK1 Q13464 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4725763 0.83 AKT1 (0.64) AKT1LIMK1ROCK2PRKACAPRKACG
SCHEMBL4726055 0.81 AKT1 (0.60) AKT1LIMK1ROCK2PRKACAPRKACG
SCHEMBL4796846 0.80 AKT1 (0.63) AKT1
SCHEMBL4778662 0.79 AKT1 (0.62) AKT1LIMK1ROCK2PRKACAPRKACG
SCHEMBL4726082 0.78 AKT1 (0.70) AKT1LIMK1ROCK2PRKACAPRKACG
SCHEMBL4727205 0.78 AKT1 (0.73) AKT1LIMK1ROCK2PRKACAPRKACG
SCHEMBL4918784 0.75 AKT1 (0.73) AKT1LIMK1ROCK2PRKACAPRKACG
SCHEMBL4778792 0.74 AKT1 (0.64) AKT1LIMK2
SCHEMBL4776438 0.74 AKT1 (0.64) AKT1LIMK1ROCK2PRKACAPRKACG
SCHEMBL4776369 0.73 AKT1 (0.61) AKT1LIMK1ROCK2PRKACAPRKACG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008012635-A2 AMINE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 2008-01-31 WO disclosed