SCHEMBL4782250

SCHEMBL4782250

COc1ccc(-c2cc3ccncc3[nH]2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.63
NPC1 O15118 3/20 0.63
RAB9A P51151 3/20 0.63
MAPT P10636 3/20 0.63
CASP3 P42574 1/20 0.63
SENP8 Q96LD8 1/20 0.63
SENP7 Q9BQF6 1/20 0.63
SENP6 Q9GZR1 1/20 0.63
CCNB2 O95067 2/20 0.57
CDK1 P06493 2/20 0.57
CCNB1 P14635 2/20 0.57
CCNB3 Q8WWL7 2/20 0.57
RIPK1 Q13546 1/20 0.57
GSK3A P49840 1/20 0.52
GSK3B P49841 1/20 0.52
CDK5 Q00535 1/20 0.52
CDK5R1 Q15078 1/20 0.52
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CHUK O15111 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21565947 0.98 KDM4E (0.61) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL14115608 0.88 KDM4E (0.63) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL26670160 0.84 CYP19A1 (0.47) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL21566048 0.83 CLK2 (0.52) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL21565988 0.82 CYP19A1 (0.50) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL27075650 0.82 CYP19A1 (0.53) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL22021633 0.81 NPY5R (0.51) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL21566047 0.80 CYP19A1 (0.47) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL6282533 0.79 KDM4E (0.47) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL7945775 0.79 KDM4E (0.73) KDM4ENPC1RAB9AMAPTCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008022467-A1 2-SUBSTITUTED AZAIN DOLES AND 2 SUBSTITUTED THIENOPYRROLES, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2008-02-28 WO disclosed
WO-2008022467-A1 2-SUBSTITUTED AZAIN DOLES AND 2 SUBSTITUTED THIENOPYRROLES, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2008-02-28 WO disclosed