SCHEMBL4782397

SCHEMBL4782397

OCC1c2ccccc2CCN1c1nc(-c2cccc(O)c2)nc(N2CCC(O)C2)n1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.39
MTOR P42345 4/20 0.36
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
IDH2 P48735 1/20 0.34
PFKFB3 Q16875 1/20 0.34
IRAK1 P51617 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
P2RY12 Q9H244 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782625 0.90 PIK3CA (0.40) PIK3CAMTORESR1ESR2PFKFB3
SCHEMBL4782618 0.90 PIK3CA (0.40) PIK3CAMTORESR1ESR2PFKFB3
SCHEMBL4884094 0.89 PIK3CA (0.44) PIK3CAMTORESR1ESR2PFKFB3
SCHEMBL4784160 0.89 PIK3CA (0.42) PIK3CAMTORESR1ESR2PFKFB3
SCHEMBL4784132 0.88 PIK3CA (0.44) PIK3CAMTORESR1ESR2PFKFB3
SCHEMBL4785045 0.86 PIK3CA (0.39) PIK3CAMTORESR1ESR2IDH2
SCHEMBL4785055 0.86 PIK3CA (0.39) PIK3CAMTORESR1ESR2IDH2
SCHEMBL4785307 0.86 PIK3CA (0.40) PIK3CAMTORESR1ESR2PFKFB3
SCHEMBL4785552 0.86 PIK3CA (0.42) PIK3CAMTORESR1ESR2PFKFB3
SCHEMBL4783923 0.86 HRH4 (0.43) PIK3CAMTORESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed