SCHEMBL4782775

SCHEMBL4782775

COc1ccc2nc(-c3n[nH]cc3C=Cc3cccnc3)[nH]c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.69
AURKA O14965 6/20 0.69
ERBB2 P04626 4/20 0.52
NPC1 O15118 5/20 0.47
RAB9A P51151 4/20 0.47
TP53 P04637 3/20 0.47
HPGD P15428 3/20 0.47
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
HSD17B10 Q99714 1/20 0.47
RUNX1 Q01196 1/20 0.47
PDPK1 O15530 1/20 0.45
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782770 1.00 KDR (0.69) KDRAURKAERBB2NPC1RAB9A
SCHEMBL13596389 0.88 KDR (0.68) KDRAURKAERBB2NPC1RAB9A
SCHEMBL4781712 0.88 KDR (0.68) KDRAURKAERBB2NPC1RAB9A
SCHEMBL13596385 0.85 KDR (0.68) KDRAURKAERBB2NPC1RAB9A
SCHEMBL14223421 0.83 KDR (0.59) KDRAURKAERBB2NPC1RAB9A
SCHEMBL13596384 0.83 KDR (0.48) KDRAURKAERBB2NPC1RAB9A
SCHEMBL13596386 0.83 KDR (0.48) KDRAURKAERBB2NPC1RAB9A
SCHEMBL13596387 0.82 KDR (0.71) KDRAURKAERBB2NPC1RAB9A
SCHEMBL13596388 0.82 KDR (0.69) KDRAURKAERBB2NPC1RAB9A
SCHEMBL4783686 0.82 KDR (0.69) KDRAURKAERBB2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048502-A1 SUBSTITUTED PYRAZOLE KINASE INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2008-04-24 WO disclosed