SCHEMBL4782873

SCHEMBL4782873

Cc1nc(=O)c(C(=O)NCC(=O)O)c(O)n1C1CCCCC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 7/20 0.63
HIF1AN Q9NWT6 2/20 0.63
OGFOD1 Q8N543 1/20 0.63
EGLN2 Q96KS0 1/20 0.63
EGLN3 Q9H6Z9 1/20 0.63
BBOX1 O75936 1/20 0.41
ASPH Q12797 1/20 0.41
KDM8 Q8N371 1/20 0.41
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
CNR2 P34972 1/20 0.38
GAA P10253 1/20 0.38
ALOX15 P16050 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
APEX1 P27695 1/20 0.38
OGFRL1 Q5TC84 2/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739996 0.86 EGLN1 (0.61) EGLN1HIF1ANOGFOD1EGLN2EGLN3
SCHEMBL4993693 0.83 EGLN1 (0.63) EGLN1HIF1ANOGFOD1EGLN2EGLN3
SCHEMBL3422098 0.78 EGLN1 (1.00) EGLN1HIF1ANOGFOD1EGLN2EGLN3
SCHEMBL1641734 0.78 EGLN1 (0.77) EGLN1HIF1ANOGFOD1EGLN2EGLN3
SCHEMBL3419112 0.78 EGLN1 (1.00) EGLN1HIF1ANOGFOD1EGLN2EGLN3
SCHEMBL3421361 0.78 EGLN1 (1.00) EGLN1HIF1ANOGFOD1EGLN2EGLN3
SCHEMBL3423522 0.78 EGLN1 (1.00) EGLN1HIF1ANOGFOD1EGLN2EGLN3
SCHEMBL3422096 0.78 EGLN1 (1.00) EGLN1HIF1ANOGFOD1EGLN2EGLN3
SCHEMBL3423425 0.77 EGLN1 (0.97) EGLN1HIF1ANOGFOD1EGLN2EGLN3
Bicarbonate SCHEMBL15419071 0.77 EGLN1 (0.97) EGLN1HIF1ANOGFOD1EGLN2EGLN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008089051-A1 N-SUBSTITUTED GLYCINE DERIVATIVES: PROLYL HYDROXYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-24 WO disclosed