SCHEMBL4787118

SCHEMBL4787118

CCOC(=O)CCNc1nc(OC)c(NC(=O)c2csc(Oc3cc(C(C)(C)C)ccc3C)n2)c(OC)n1.Cc1ccc(C(C)(C)C)cc1Oc1nc(C(=O)O)cs1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.35
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GNRHR P30968 2/20 0.32
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
CACNA1F O60840 1/20 0.31
CHRM4 P08173 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
CHRM1 P11229 1/20 0.31
CYP2C9 P11712 1/20 0.31
DRD1 P21728 1/20 0.31
DRD4 P21917 1/20 0.31
SLC6A2 P23975 1/20 0.31
HRH2 P25021 1/20 0.31
TACR1 P25103 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4233364 0.97 TOP2A (0.35) TOP2ALMNANPSR1HSD17B10NPC1
SCHEMBL4228796 0.90 KDM4E (0.35) LMNANPSR1HSD17B10GNRHRHPGD
SCHEMBL13743595 0.89 GNRHR (0.34) LMNANPSR1HSD17B10GNRHRHPGD
SCHEMBL13743435 0.89 GNRHR (0.35) LMNANPSR1HSD17B10GNRHRHPGD
SCHEMBL4237338 0.88 GNRHR (0.34) LMNANPSR1HSD17B10GNRHRCACNA1F
SCHEMBL4236457 0.88 SYK (0.36) GNRHRHPGDTSHRCACNA1FCHRM4
SCHEMBL4685725 0.88 GNRHR (0.32) GNRHRCACNA1FCHRM4ADORA3CHRM1
SCHEMBL4226409 0.87 IRAK4 (0.35) GNRHRHPGDCACNA1FCHRM4ADORA3
SCHEMBL4233435 0.86 GNRHR (0.35) LMNANPSR1HSD17B10GNRHRCACNA1F
SCHEMBL4231634 0.86 GNRHR (0.42) LMNANPC1RAB9ASMN1; SMN2GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896465-A1 HETEROCYCLIC NON-PEPTIDE GNRH ANTAGONISTS Takeda Cambridge Limited (GB) 2008-03-12 EP disclosed
WO-2007000582-A1 HETEROCYCLIC NON-PEPTIDE GNRH ANTAGONISTS TAKEDA CAMBRIDGE LIMITED (GB) 2007-01-04 WO disclosed