SCHEMBL4788009

SCHEMBL4788009

O=C(NC1CCCCC1)[C@H](C1CCCCC1)n1c(-c2ccc(-c3nnn[nH]3)cc2)nc2ccccc21

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.72
KCNH2 Q12809 4/20 0.54
CYP3A4 P08684 3/20 0.54
CYP2D6 P10635 2/20 0.54
CYP2C9 P11712 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788026 1.00 NR1H4 (0.72) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL3558696 0.99 NR1H4 (0.71) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL3558693 0.98 NR1H4 (0.71) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL3565567 0.91 NR1H4 (0.64) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL3565563 0.91 NR1H4 (0.65) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL3573957 0.86 NR1H4 (0.86) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL3557195 0.85 NR1H4 (0.84) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL3571353 0.84 NR1H4 (0.81) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL3572739 0.84 NR1H4 (0.81) NR1H4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL3565319 0.84 NR1H4 (1.00) NR1H4KCNH2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008155054-A1 FARNESOID-X-RECEPTOR MUTANTS, AND CRYSTALLISATION THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2008-12-24 WO disclosed