SCHEMBL4789585

SCHEMBL4789585

CC1CN(c2ccncc2)CCN1c1nc(-c2ccncc2)cc(=O)n1C

nearest known ligand 0.78

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.78
CYP2D6 P10635 11/20 0.68
CYP1A2 P05177 8/20 0.66
CYP3A4 P08684 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL698099 1.00 GSK3B (0.78) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL703251 0.93 GSK3B (0.70) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL698296 0.93 GSK3B (0.78) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL698132 0.93 GSK3B (0.70) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL8235407 0.92 GSK3B (0.79) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL698110 0.91 GSK3B (0.78) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL695864 0.90 GSK3B (0.79) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL696557 0.90 GSK3B (0.67) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL700672 0.88 GSK3B (0.78) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL695353 0.88 GSK3B (0.78) GSK3BCYP2D6CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001863-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS Mitsubishi Tanabe Pharma Corporation (JP) 2008-12-17 EP disclosed
WO-2007119463-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-10-25 WO disclosed
WO-2007119463-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-10-25 WO disclosed