SCHEMBL4789893

SCHEMBL4789893

C[C@H]1CC[C@H](C(=O)N(CC(F)F)c2cc(-c3ccc(-c4cc5ncccn5n4)cc3)sc2C(=O)O)CC1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.36
APOBEC3A P31941 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
PDE4D Q08499 2/20 0.32
OPRM1 P35372 1/20 0.31
SYK P43405 1/20 0.31
NR1I2 O75469 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4789894 1.00 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GPDE4DOPRM1
SCHEMBL4824071 0.93 KDM4E (0.36) PDE4DSYK
SCHEMBL4824077 0.93 KDM4E (0.36) PDE4DSYK
SCHEMBL4815926 0.92 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GOPRM1NR1I2
SCHEMBL4838993 0.91 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GSYKNR1I2
SCHEMBL4838987 0.91 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GSYKNR1I2
Ammonia Solution, Strong SCHEMBL4156140 0.90 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GSYKNR1I2
Ammonia Solution, Strong SCHEMBL4156138 0.90 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GSYKNR1I2
SCHEMBL4823086 0.89 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GPDE4DSYK
SCHEMBL4823092 0.89 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GPDE4DSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000818-A1 3-CARBONYLAMINOTHIOPHENE-2-CARBOXYLIC ACIDS AS HEPATITIS C VIRUS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-31 WO claimed
WO-2009000818-A1 3-CARBONYLAMINOTHIOPHENE-2-CARBOXYLIC ACIDS AS HEPATITIS C VIRUS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-31 WO disclosed
WO-2009000818-A1 3-CARBONYLAMINOTHIOPHENE-2-CARBOXYLIC ACIDS AS HEPATITIS C VIRUS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-31 WO disclosed