SCHEMBL4790334

SCHEMBL4790334

Cc1nnc(N2CCC(N3COc4cccnc43)CC2)n1-c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 14/20 0.46
OXTR P30559 8/20 0.37
TRPA1 O75762 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.36
CHI3L1 P36222 1/20 0.35
KCNH2 Q12809 1/20 0.35
CHIT1 Q13231 1/20 0.35
CHI3L2 Q15782 1/20 0.35
CHIA Q9BZP6 1/20 0.35
AVPR1B P47901 1/20 0.34
BRD4 O60885 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
USP14 P54578 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4713503 0.91 AVPR1A (0.45) AVPR1AOXTRTRPA1TRPM8CHI3L1
SCHEMBL4710762 0.84 AVPR1A (0.43) AVPR1AOXTRTRPA1TRPM8CHI3L1
SCHEMBL4760978 0.74 AVPR1A (0.47) AVPR1AOXTRTRPA1TRPM8
SCHEMBL4714355 0.74 AVPR1A (0.47) AVPR1AOXTRTRPA1TRPM8KCNH2
SCHEMBL4712455 0.74 AVPR1A (0.44) AVPR1AOXTRTRPA1TRPM8KCNH2
SCHEMBL5436364 0.73 AVPR1A (0.53) AVPR1AOXTRTRPA1TRPM8
SCHEMBL5426182 0.73 AVPR1A (0.54) AVPR1AOXTRTRPA1TRPM8BRD4
SCHEMBL5428048 0.73 AVPR1A (0.52) AVPR1AOXTRTRPA1TRPM8DRD3
SCHEMBL4713593 0.72 AVPR1A (0.45) AVPR1AOXTRKCNH2DRD4DRD3
SCHEMBL5155966 0.72 AVPR1A (0.48) AVPR1AOXTRTRPA1TRPM8BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877399-A1 TRIAZOLE DERIVATIVES AS VASOPRESSIN ANTAGONISTS Pfizer Limited (GB) 2008-01-16 EP claimed
WO-2006114706-A1 TRIAZOLE DERIVATIVES AS VASOPRESSIN ANTAGONISTS PFIZER LIMITED (GB) 2006-11-02 WO claimed