SCHEMBL4791

SCHEMBL4791

Cc1noc(-c2ccc(-c3ccc(C4(CC(=O)O)CC4)cc3)cc2)c1NCCc1cc(-c2ccccc2)no1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
MAPT P10636 3/20 0.42
LMNA P02545 2/20 0.42
POLB P06746 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
LPAR1 Q92633 4/20 0.41
ABCC3 O15438 1/20 0.41
ABCC4 O15439 1/20 0.41
ABCB11 O95342 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2C9 P11712 1/20 0.41
ABCB4 P21439 1/20 0.41
ABCC2 Q92887 1/20 0.41
SLCO1B3 Q9NPD5 1/20 0.41
SLCO1B1 Q9Y6L6 1/20 0.41
IGF1R P08069 1/20 0.38
MMP2 P08253 2/20 0.38
MMP8 P22894 2/20 0.38
MMP12 P39900 2/20 0.38
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4090 0.91 LPAR1 (0.40) ALDH1A1MAPTLMNAPOLBRXFP1
SCHEMBL7223 0.83 LPAR1 (0.41) ALDH1A1MAPTLPAR1ABCC3ABCC4
SCHEMBL13530 0.82 LPAR1 (0.45) ALDH1A1MAPTLMNAPOLBRXFP1
SCHEMBL6412 0.81 LPAR1 (0.40) ALDH1A1MAPTLPAR1ABCC3ABCC4
SCHEMBL4348 0.80 IGF1R (0.43) ALDH1A1MAPTLMNAPOLBRXFP1
SCHEMBL3954 0.79 LPAR1 (0.43) ALDH1A1MAPTLMNAPOLBRXFP1
SCHEMBL4790 0.75 BRD4 (0.34) ALDH1A1MAPTLMNAPOLBRXFP1
SCHEMBL13437 0.74 LPAR1 (0.44) ALDH1A1MAPTLPAR1ABCC3ABCC4
SCHEMBL10387 0.74 LPAR1 (0.47) ALDH1A1MAPTLPAR1ABCC3ABCC4
SCHEMBL6642 0.73 LPAR1 (0.39) MAPTLPAR1ABCC3ABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP claimed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO claimed
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed