SCHEMBL4794802

SCHEMBL4794802

C#CCn1c(=O)c2c(nc(C#Cc3cccc(OCc4ccccc4)c3)n2C)n(C)c1=O

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.47
MAOB P27338 4/20 0.47
ADORA2A P29274 3/20 0.47
ADORA2B P29275 1/20 0.46
MAOA P21397 2/20 0.45
PKM P14618 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4952866 0.89 ADORA1 (0.42) ADORA1MAOBADORA2AADORA2BMAOA
SCHEMBL2536366 0.89 ADORA1 (0.47) ADORA1MAOBADORA2AADORA2BMAOA
SCHEMBL2537627 0.87 ADORA1 (0.57) ADORA1MAOBADORA2AADORA2B
SCHEMBL2542698 0.87 ADORA1 (0.47) ADORA1MAOBADORA2AADORA2B
SCHEMBL2537641 0.87 ADORA2A (0.46) ADORA1MAOBADORA2AADORA2B
SCHEMBL2537917 0.86 ADORA1 (0.45) ADORA1MAOBADORA2AADORA2B
SCHEMBL2541481 0.86 ADORA2A (0.49) ADORA1MAOBADORA2AADORA2B
SCHEMBL2535874 0.85 ADORA1 (0.45) ADORA1MAOBADORA2AADORA2B
SCHEMBL2541195 0.85 ADORA2A (0.52) ADORA1MAOBADORA2AADORA2B
SCHEMBL2541035 0.85 ADORA1 (0.47) ADORA1MAOBADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed