SCHEMBL4796196

SCHEMBL4796196

CS(=O)(=O)Cc1nc(N2CC(C(=O)NS(=O)(=O)Cc3ccccc3)C2)c(C#N)cc1C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 19/20 0.69
CYP3A4 P08684 4/20 0.59
CYP2C9 P11712 3/20 0.59
CHRM2 P08172 1/20 0.58
DRD3 P35462 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4891753 0.90 P2RY12 (0.82) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL3217388 0.89 P2RY12 (0.82) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL3589485 0.84 P2RY12 (0.70) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL3226299 0.83 P2RY12 (0.80) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4873260 0.83 P2RY12 (0.85) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL3327629 0.83 P2RY12 (0.84) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4783399 0.82 P2RY12 (0.83) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL3325916 0.82 P2RY12 (0.82) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL3590558 0.82 P2RY12 (0.82) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4740602 0.82 P2RY12 (0.71) P2RY12CYP3A4CYP2C9CHRM2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008085119-A1 NEW PYRIDINE ANALOGUES VIII 518 ASTRAZENECA AB (SE) 2008-07-17 WO disclosed