SCHEMBL4796398

SCHEMBL4796398

COC(=O)c1sc(I)cc1N(C(=O)C1CCC(C)CC1)C1CCOC1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
RAB9A P51151 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HSD17B10 Q99714 1/20 0.33
NR1I2 O75469 2/20 0.32
CYP2E1 P05181 1/20 0.31
HTT P42858 1/20 0.30
ATM Q13315 1/20 0.30
NPC1 O15118 1/20 0.30
HSP90AA1 P07900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4796389 1.00 KDM4E (0.33) KDM4ERAB9AALDH1A1HSD17B10NR1I2
SCHEMBL14290668 0.94 CYP2E1 (0.34) KDM4ERAB9AALDH1A1HSD17B10NR1I2
SCHEMBL2432624 0.91 NR1I2 (0.32) KDM4EALDH1A1NR1I2CYP2E1HTT
SCHEMBL2432640 0.91 NR1I2 (0.32) KDM4EALDH1A1NR1I2CYP2E1HTT
SCHEMBL938959 0.88 KDM4E (0.30) KDM4ERAB9AALDH1A1HSD17B10
SCHEMBL12909947 0.88 KDM4E (0.30) KDM4ERAB9AALDH1A1HSD17B10
SCHEMBL2432488 0.87 NR1I2 (0.36) KDM4ERAB9AALDH1A1HSD17B10NR1I2
SCHEMBL2432492 0.87 NR1I2 (0.36) KDM4ERAB9AALDH1A1HSD17B10NR1I2
SCHEMBL102056 0.85 NR1I2 (0.33) KDM4ERAB9AALDH1A1NR1I2HTT
SCHEMBL139451 0.85 NR1I2 (0.33) KDM4ERAB9AALDH1A1NR1I2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed