SCHEMBL4796693

SCHEMBL4796693

COc1cccc(CC(Cc2ccccc2)Nc2nnc(-c3ccc4cnccc4c3)s2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 5/20 0.50
PRKACA P17612 4/20 0.50
AKT1 P31749 2/20 0.47
CDK2 P24941 2/20 0.47
SGK1 O00141 1/20 0.47
DYRK1A Q13627 1/20 0.44
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
NOX1 Q9Y5S8 2/20 0.40
ROCK2 O75116 2/20 0.40
KDM4E B2RXH2 3/20 0.39
HSD17B10 Q99714 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CDC7 O00311 1/20 0.39
CCNE1 P24864 1/20 0.39
DBF4 Q9UBU7 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
ESR1 P03372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4850255 0.92 ROCK1 (0.49) ROCK1PRKACAAKT1CDK2SGK1
SCHEMBL4781794 0.87 ROCK1 (0.45) ROCK1PRKACAAKT1CDK2SGK1
SCHEMBL4890207 0.85 AKT1 (0.52) ROCK1PRKACAAKT1CDK2SGK1
SCHEMBL4899252 0.84 AKT1 (0.53) ROCK1AKT1CDK2SGK1NOX1
SCHEMBL4898277 0.84 AKT1 (0.53) ROCK1AKT1CDK2SGK1NOX1
SCHEMBL4780577 0.84 AKT1 (0.53) ROCK1AKT1CDK2SGK1NOX1
SCHEMBL4779887 0.84 AKT1 (0.49) ROCK1PRKACAAKT1CDK2SGK1
SCHEMBL4890399 0.83 AKT1 (0.52) ROCK1AKT1CDK2SGK1NOX1
SCHEMBL4902138 0.83 AKT1 (0.52) ROCK1AKT1CDK2SGK1NOX1
SCHEMBL4898250 0.83 AKT1 (0.52) ROCK1AKT1CDK2SGK1NOX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008036308-A2 AMINO-SUBSTITUTED HETEROCYCLES, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2008-03-27 WO disclosed