SCHEMBL4797977

SCHEMBL4797977

NS(=O)(=O)c1ccc([AsH]c2nc(Nc3ccc4[nH]ncc4c3)nc3[nH]ncc23)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.58
CCNT1 O60563 2/20 0.46
CDK1 P06493 2/20 0.46
CCNB1 P14635 2/20 0.46
CDK2 P24941 2/20 0.46
CDK7 P50613 2/20 0.46
CDK9 P50750 2/20 0.46
CCNH P51946 2/20 0.46
CDK5 Q00535 1/20 0.46
MKNK1 Q9BUB5 1/20 0.45
CDC7 O00311 1/20 0.41
MAPK1 P28482 1/20 0.41
LYN P07948 1/20 0.41
TXK P42681 1/20 0.41
SYK P43405 1/20 0.41
BTK Q06187 1/20 0.41
CA1 P00915 5/20 0.40
CA2 P00918 5/20 0.40
CA9 Q16790 5/20 0.40
CA12 O43570 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4267261 0.84 KDR (0.64) KDRCCNT1CDK1CCNB1CDK2
SCHEMBL13896206 0.74 CCNT1 (0.58) KDRCCNT1CDK1CCNB1CDK2
SCHEMBL31647068 0.73 KDR (0.57) KDRCDK5MAPK1ROCK1
SCHEMBL5220947 0.73 KDR (0.57) KDRCDK5MAPK1ROCK1
SCHEMBL13896209 0.72 MKNK1 (0.67) KDRCDK2MKNK1CDC7SYK
SCHEMBL4266513 0.70 PLK4 (0.57) KDRCCNT1CDK1CCNB1CDK2
SCHEMBL13896208 0.70 PLK4 (0.57) KDRCCNT1CDK1CCNB1CDK2
SCHEMBL6081930 0.70 KDR (0.59) KDRCCNT1CDK1CCNB1CDK2
SCHEMBL10242647 0.70 SYK (0.67) KDRCCNT1CDK1CCNB1CDK2
SCHEMBL3283879 0.69 KDR (0.50) KDRCCNT1CDK1CCNB1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008039359-A2 BICYCLIC PYRIMIDINE KINASE INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2008-04-03 WO claimed