SCHEMBL4800201

SCHEMBL4800201

COC(=O)c1cccc(-c2ccc3c(c2)/C=C\c2ccccc2N(C(C)=O)C3)n1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 7/20 0.43
FAAH O00519 6/20 0.40
SCN9A Q15858 3/20 0.39
P2RX4 Q99571 1/20 0.36
BCL2L1 Q07817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6388516 0.89 HSD17B3 (0.46) HSD17B3SCN9ABCL2L1
SCHEMBL6388510 0.89 HSD17B3 (0.46) HSD17B3SCN9ABCL2L1
SCHEMBL4797023 0.88 HSD17B3 (0.43) HSD17B3SCN9ABCL2L1
SCHEMBL4797028 0.88 HSD17B3 (0.43) HSD17B3SCN9ABCL2L1
SCHEMBL4799309 0.86 HSD17B3 (0.45) HSD17B3
SCHEMBL4799318 0.86 HSD17B3 (0.45) HSD17B3
SCHEMBL4798174 0.83 HSD17B3 (0.46) HSD17B3SCN9A
SCHEMBL4798186 0.83 HSD17B3 (0.46) HSD17B3SCN9A
SCHEMBL4804464 0.81 HSD17B3 (0.39) HSD17B3P2RX4
SCHEMBL4804473 0.81 HSD17B3 (0.39) HSD17B3P2RX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7417040-B2 Fused tricyclic compounds as inhibitors of 17β-hydroxysteroid dehydrogenase 3 BRISTOL-MYERS SQUIBB COMPANY (US) 2008-08-26 US disclosed