SCHEMBL4800631

SCHEMBL4800631

CC(=O)NC1CN(c2nc3c(C#N)c(C)c(-c4ccccc4)c(N4CC[C@H](N(C)C)C4)c3o2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 4/20 0.38
MCHR1 Q99705 4/20 0.35
CKS1B P61024 1/20 0.35
SKP1 P63208 1/20 0.35
SKP2 Q13309 1/20 0.35
MAPK8 P45983 2/20 0.35
BTK Q06187 2/20 0.35
MRGPRX2 Q96LB1 2/20 0.35
MAPK10 P53779 1/20 0.35
BCL6 P41182 1/20 0.35
HTR1D P28221 2/20 0.34
HTR3A P46098 2/20 0.34
HTR6 P50406 2/20 0.34
TMEM97 Q5BJF2 2/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
HTR1B P28222 1/20 0.34
SLC6A3 Q01959 1/20 0.34
ADRA1B P35368 1/20 0.34
CTSL P07711 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3296758 0.96 MCHR1 (0.37) MCHR1MAPK8BTKMRGPRX2MAPK10
SCHEMBL3297399 0.90 MCHR1 (0.38) MCHR1MAPK8BTKMRGPRX2MAPK10
SCHEMBL3300554 0.90 MCHR1 (0.36) MCHR1MAPK8BTKMRGPRX2MAPK10
SCHEMBL3299211 0.88 KDM4E (0.37) MCHR1MAPK8BTKMRGPRX2MAPK10
SCHEMBL3295055 0.88 HTR1D (0.37) MCHR1MAPK8BTKMRGPRX2MAPK10
SCHEMBL3295295 0.88 HTR1D (0.34) MCHR1MAPK8BTKMRGPRX2MAPK10
SCHEMBL3293642 0.87 KHK (0.36) MCHR1MAPK8BTKMRGPRX2MAPK10
SCHEMBL4800625 0.87 SMPD3 (0.35) SMPD3CKS1BSKP1SKP2LRRK2
SCHEMBL3295980 0.86 HTR1D (0.38) MAPK8BTKMRGPRX2MAPK10HTR1D
SCHEMBL3294312 0.86 HTR1D (0.38) MAPK8BTKMRGPRX2MAPK10HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1932837-A1 BICYCLO HETEROCYCLIC COMPOUND HAVING ANTIFUNGAL ACTION Daiichi Sankyo Company, Limited (JP) 2008-06-18 EP disclosed