SCHEMBL480143

SCHEMBL480143

Cc1cc(C(C)(O)Cc2ccc(Oc3ccc(C#N)cc3)cc2Cl)ccn1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.38
KCNH2 Q12809 2/20 0.38
GRM2 Q14416 4/20 0.37
SCN9A Q15858 3/20 0.37
SLC6A4 P31645 1/20 0.36
GRM5 P41594 1/20 0.35
NR3C2 P08235 2/20 0.35
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
CYP19A1 P11511 1/20 0.33
KDR P35968 1/20 0.32
GCK P35557 1/20 0.32
PTGER4 P35408 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480120 0.75 AR (0.38) GRM2SCN9AGRM5CYP11B1CYP11B2
SCHEMBL30689353 0.73 CYP19A1 (0.49) KCNH2GRM2SCN9AGRM5CYP19A1
SCHEMBL479812 0.68 HTR2A (0.47) HTR2AKCNH2SCN9ASLC6A4PGR
SCHEMBL479920 0.68 SCN9A (0.36) HTR2AKCNH2GRM2SCN9ASLC6A4
SCHEMBL479759 0.67 CYP11B1 (0.40) KCNH2GRM2SCN9ACYP11B1CYP11B2
SCHEMBL14833394 0.64 HTR2A (0.56) HTR2AKCNH2SLC6A4CYP11B1CYP11B2
SCHEMBL9889460 0.64 HTR2A (0.46) HTR2AKCNH2SLC6A4CYP19A1
SCHEMBL22349702 0.63 AR (0.46) HTR2AKCNH2SCN9ASLC6A4CYP19A1
SCHEMBL922673 0.63 HTR2A (0.52) HTR2AKCNH2SLC6A4PGR
SCHEMBL3700809 0.62 KCNH2 (0.49) HTR2AKCNH2SCN9ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed