Bromide

Bromide

SCHEMBL4811327

Br.CCCCc1cc(C(=O)CN2Cc3cc(OCC)c(C(=O)NC)cc3C2=N)cc(N(C)C)c1O

nearest known ligand 0.34

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
F2R P25116 6/20 0.33
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
CRHBP P24387 1/20 0.31
KMT2A Q03164 1/20 0.31
CRHR2 Q13324 1/20 0.31
HIF1A Q16665 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL1728975 0.86 F2R (0.42) KDM4ENPC1MAPTRAB9AF2R
SCHEMBL14449104 0.85 F2R (0.41) KDM4ENPC1MAPTRAB9AF2R
Bromide SCHEMBL5488732 0.85 KDM4E (0.35) KDM4ENPC1MAPTRAB9AF2R
Bromide SCHEMBL6544809 0.85 F2R (0.37) KDM4ENPC1MAPTRAB9AF2R
Bromide SCHEMBL1731380 0.83 KDM4E (0.34) KDM4ENPC1MAPTRAB9AF2R
Hydrochloric Acid SCHEMBL1729535 0.83 MAPT (0.38) KDM4ENPC1MAPTRAB9AF2R
Bromide SCHEMBL1729646 0.81 F2R (0.48) KDM4ENPC1MAPTRAB9AF2R
Bromide SCHEMBL1729603 0.81 F2R (0.40) KDM4ENPC1MAPTRAB9AF2R
Bromide SCHEMBL1730337 0.81 F2R (0.40) KDM4ENPC1MAPTRAB9AF2R
Bromide SCHEMBL1731536 0.80 F2R (0.43) KDM4ENPC1MAPTRAB9AF2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008128038-A2 METHODS AND COMPOSITIONS FOR TREATING CARDIAC DYSFUNCTIONS THE SCRIPPS RESEARCH INSTITUTE (US) 2008-10-23 WO claimed