SCHEMBL4819965

SCHEMBL4819965

COc1cc2nccc(Oc3ccc4c(c3)OCCN4C(=O)NN(C)C)c2cc1OC

nearest known ligand 0.82

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDR P35968 20/20 0.82
LCK P06239 17/20 0.82
MET P08581 16/20 0.79
TEK Q02763 12/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4548979 0.90 KDR (1.00) KDRLCKMETTEK
SCHEMBL2746417 0.89 KDR (0.84) KDRLCKMETTEK
SCHEMBL2748661 0.88 KDR (1.00) KDRLCKMETTEK
SCHEMBL4548970 0.88 KDR (1.00) KDRLCKMETTEK
SCHEMBL2747939 0.87 KDR (1.00) KDRLCKMETTEK
SCHEMBL2748420 0.87 KDR (1.00) KDRLCKMETTEK
SCHEMBL2747312 0.86 KDR (1.00) KDRLCKMETTEK
SCHEMBL2747431 0.86 KDR (1.00) KDRLCKMETTEK
SCHEMBL2747171 0.86 KDR (0.79) KDRLCKMETTEK
SCHEMBL4548981 0.85 KDR (0.77) KDRLCKMETTEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435823-B2 Compounds and methods of use AMGEN INC. (US) 2008-10-14 US claimed