SCHEMBL4823324

SCHEMBL4823324

COC(=O)[C@H](Cc1ccc(-c2ccc(Cl)cc2)cc1)NC(=O)c1cc2ccccc2cc1O

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.56
KDR P35968 1/20 0.56
HDAC1 Q13547 6/20 0.52
HDAC6 Q9UBN7 6/20 0.52
PYGL P06737 1/20 0.52
TACR3 P29371 1/20 0.51
NOS2 P35228 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4823322 1.00 CDK2 (0.56) CDK2KDRHDAC1HDAC6PYGL
SCHEMBL13986736 0.93 KDR (0.60) CDK2KDRHDAC1HDAC6TACR3
SCHEMBL4824089 0.93 KDR (0.60) CDK2KDRHDAC1HDAC6TACR3
SCHEMBL4824091 0.93 KDR (0.60) CDK2KDRHDAC1HDAC6TACR3
SCHEMBL4827846 0.90 HDAC1 (0.63) CDK2KDRHDAC1HDAC6TACR3
SCHEMBL4827850 0.90 HDAC1 (0.63) CDK2KDRHDAC1HDAC6TACR3
SCHEMBL4824679 0.90 KDR (0.51) CDK2KDRHDAC1HDAC6PYGL
SCHEMBL4824673 0.90 KDR (0.51) CDK2KDRHDAC1HDAC6PYGL
SCHEMBL4829720 0.89 KDR (0.56) CDK2KDRHDAC1HDAC6TACR3
SCHEMBL4829713 0.89 KDR (0.56) CDK2KDRHDAC1HDAC6TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7459472-B2 Aryl and heteroaryl compounds, compositions, and methods of use TRANSTECH PHARMA, INC. (US) 2008-12-02 US disclosed
US-20050059713-A1 Aryl and heteroaryl compounds, compositions, and methods of use VTVX HOLDINGS I LLC 2005-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050059713-A1 Aryl and heteroaryl compounds, compositions, and methods of use CYP2F1, CYP3A43, PNPO CDK2 456/4885KDR 1624/4885HDAC1 1171/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.