SCHEMBL483619

SCHEMBL483619

COC(=O)[C@H]1CCC(c2ccc(OCc3ccccc3)cc2)=N1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
NPC1 O15118 2/20 0.47
NR4A1 P22736 1/20 0.47
NR4A2 P43354 1/20 0.47
NR4A3 Q92570 1/20 0.47
MAOB P27338 1/20 0.45
ACACB O00763 1/20 0.45
ALDH1A1 P00352 1/20 0.44
GSK3B P49841 1/20 0.44
BACE1 P56817 1/20 0.44
SRD5A2 P31213 1/20 0.44
KDM4E B2RXH2 2/20 0.43
KMT2A Q03164 2/20 0.43
FFAR1 O14842 1/20 0.42
MEN1 O00255 1/20 0.42
PABPC1 P11940 1/20 0.42
SMPD1 P17405 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17873425 1.00 CA1 (0.50) CA1CA2RAB9ASMN1; SMN2NPC1
SCHEMBL310921 1.00 CA1 (0.50) CA1CA2RAB9ASMN1; SMN2NPC1
SCHEMBL483661 0.89 MAPT (0.50) CA1CA2NR4A1NR4A2NR4A3
SCHEMBL13311119 0.89 MAPT (0.50) CA1CA2NR4A1NR4A2NR4A3
SCHEMBL20876895 0.88 NR4A2 (0.51) CA1CA2RAB9ANR4A1NR4A2
SCHEMBL2713179 0.88 NR4A2 (0.51) CA1CA2RAB9ANR4A1NR4A2
SCHEMBL2727830 0.88 NR4A2 (0.51) CA1CA2RAB9ANR4A1NR4A2
SCHEMBL483467 0.88 JAK2 (0.46) NR4A2MAOBSRD5A2SMPD1
SCHEMBL22534143 0.86 KCNH2 (0.50) CA1CA2RAB9ASMN1; SMN2NPC1
SCHEMBL22534142 0.86 KCNH2 (0.50) CA1CA2RAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1934176-B1 QUATERNARY ALPHA-AMINOCARBOXAMIDE DERIVATIVES AS MODULATORS OF VOLTAGE-GATED SODIUM CHANNELS GLAXO GROUP LTD (GB) 2012-02-01 EP disclosed