SCHEMBL4844745

SCHEMBL4844745

COc1cc(C)c(S(=O)(=O)C(C)CCOCC(=O)N(C)Cc2ccc(C3=NCCN3)cc2)c(C)c1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 15/20 0.75
NISCH Q9Y2I1 2/20 0.39
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14304352 0.91 BDKRB1 (0.61) BDKRB1NISCHKDM4E
Safotibant SCHEMBL1723565 0.85 BDKRB1 (1.00) BDKRB1
SCHEMBL4030095 0.83 BDKRB1 (0.74) BDKRB1NISCH
SCHEMBL12020596 0.81 BDKRB1 (0.49) BDKRB1
SCHEMBL4036844 0.79 BDKRB1 (1.00) BDKRB1NISCH
SCHEMBL4924234 0.79 BDKRB1 (0.69) BDKRB1NISCH
SCHEMBL14304935 0.79 BDKRB1 (0.48) BDKRB1
SCHEMBL4031819 0.78 BDKRB1 (0.81) BDKRB1NISCHKDM4E
SCHEMBL4036840 0.78 BDKRB1 (0.74) BDKRB1NISCH
SCHEMBL2568098 0.77 BDKRB1 (0.64) BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008002849-A2 ARYL SULFONES NEUROGEN CORPORATION (US) 2008-01-03 WO claimed