SCHEMBL4845548

SCHEMBL4845548

CCCn1c(Cc2cc(OC)c(OC)c(OC)c2)nc2c(N)nc(F)nc21

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 16/20 0.75
HSP90AB1 P08238 16/20 0.75
ERBB2 P04626 4/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852703 0.94 HSP90AA1 (0.79) HSP90AA1HSP90AB1ERBB2
SCHEMBL4845541 0.93 HSP90AA1 (0.77) HSP90AA1HSP90AB1ERBB2
SCHEMBL4844123 0.90 HSP90AA1 (0.74) HSP90AA1HSP90AB1ERBB2
SCHEMBL4847099 0.88 HSP90AA1 (0.89) HSP90AA1HSP90AB1ERBB2
SCHEMBL4850767 0.88 HSP90AA1 (0.70) HSP90AA1HSP90AB1ERBB2
SCHEMBL4854173 0.87 HSP90AA1 (0.75) HSP90AA1HSP90AB1ERBB2
SCHEMBL4853114 0.87 HSP90AA1 (0.74) HSP90AA1HSP90AB1ERBB2
SCHEMBL4850811 0.86 HSP90AA1 (0.73) HSP90AA1HSP90AB1ERBB2
SCHEMBL4854328 0.86 HSP90AA1 (1.00) HSP90AA1HSP90AB1ERBB2
SCHEMBL4848604 0.85 HSP90AA1 (0.65) HSP90AA1HSP90AB1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1335920-B1 COMPOSITIONS CONTAINING PURINE DERIVATIVES FOR BINDING TO HSP90 SLOAN KETTERING INST CANCER (US) 2013-04-03 EP disclosed
US-7439359-B2 Small molecule compositions for binding to hsp90 SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2008-10-21 US disclosed
EP-1335920-A4 SMALL MOLECULE COMPOSITIONS FOR BINDING TO HSP90 SLOAN KETTERING INSTITUTEFOR C (US) 2005-08-17 EP disclosed
US-20040102458-A1 Small molecule compositions for binding to hsp90 SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH 2004-05-27 US disclosed
EP-1335920-A2 SMALL MOLECULE COMPOSITIONS FOR BINDING TO HSP90 Sloan-Kettering Institute For Cancer Research (US) 2003-08-20 EP disclosed
WO-2002036075-A2 SMALL MOLECULE COMPOSITIONS FOR BINDING TO HSP90 SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2002-05-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040102458-A1 Small molecule compositions for binding to hsp90 HSP90AB1, ERBB2, HSP90AB2P HSP90AA1 5/4885HSP90AB1 1/4885ERBB2 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.