SCHEMBL4847255

SCHEMBL4847255

CCOC(=O)c1cc(C)cnc1NCc1ccc(OC)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.55
MAPT P10636 9/20 0.53
ALDH1A1 P00352 5/20 0.53
LMNA P02545 4/20 0.53
KDM4E B2RXH2 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
HPGD P15428 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
KMT2A Q03164 3/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
MEN1 O00255 2/20 0.48
ASPH Q12797 1/20 0.48
RIOX2 Q8IUF8 1/20 0.48
KDM8 Q8N371 1/20 0.48
VNN1 O95497 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47
ADORA1 P30542 1/20 0.47
TP53 P04637 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14195182 0.92 KDM4E (0.51) GAAMAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL4847270 0.89 GAA (0.53) GAAMAPTALDH1A1LMNAKDM4E
SCHEMBL31278029 0.82 MAPT (0.52) GAAMAPTALDH1A1LMNAKDM4E
SCHEMBL14734451 0.81 MAPT (0.51) GAAMAPTALDH1A1LMNAKDM4E
SCHEMBL30050379 0.81 MAPT (0.51) GAAMAPTALDH1A1LMNAKDM4E
SCHEMBL18168179 0.80 MAPT (0.56) GAAMAPTALDH1A1LMNAKDM4E
SCHEMBL34462331 0.79 NPSR1 (0.57) GAAMAPTALDH1A1LMNAKDM4E
SCHEMBL23782531 0.79 MAPT (0.58) GAAMAPTALDH1A1LMNAKDM4E
SCHEMBL4851862 0.79 MCHR1 (0.59) MAPTALDH1A1LMNAKDM4ETDP1
SCHEMBL20189399 0.79 MAPT (0.53) GAAMAPTALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7361760-B2 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases AVANIR PHARMACEUTICALS (US) 2008-04-22 US disclosed
US-20070191388-A1 SUBSTITUTED NAPHTHYRIDINE DERIVATIVES AS INHIBITORS OF MACROPHAGE MIGRATION INHIBITORY FACTOR AND THEIR USE IN THE TREATMENT OF HUMAN DISEASES AVANIR PHARMACEUTICALS (US) 2007-08-16 US disclosed
US-20050124604-A1 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases AVANIR PHARMACEUTICALS, INC. 2005-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070191388-A1 SUBSTITUTED NAPHTHYRIDINE DERIVATIVES AS INHIBITORS OF MACROPHAGE MIGRATION INHIBITORY FACTOR AND THEIR USE IN THE TREATMENT OF HUMAN DISEASES MIF, MSR1, SLC11A2 GAA 604/4885MAPT 4680/4885ALDH1A1 2477/4885
US-20050124604-A1 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases MIF, MSR1, SLC11A2 GAA 604/4885MAPT 4680/4885ALDH1A1 2477/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.