SCHEMBL484946

SCHEMBL484946

CC(C)(C)OC(=O)N1CCC2(CCCNC2)CC1.O=C(O)N1CCC2(CCCN(c3ccncc3)C2)CC1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 17/20 0.60
CYP2C19 P33261 10/20 0.60
HIF1A Q16665 6/20 0.60
ALDH1A1 P00352 4/20 0.60
CYP2C9 P11712 12/20 0.56
CYP2D6 P10635 9/20 0.56
CYP1A2 P05177 7/20 0.56
TSHR P16473 6/20 0.56
ALOX15 P16050 2/20 0.56
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
USP2 O75604 5/20 0.50
MAPK1 P28482 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.47
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL484568 0.88 CYP3A4 (0.77) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
SCHEMBL484571 0.83 CYP3A4 (0.70) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
SCHEMBL485072 0.82 CYP3A4 (0.67) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
Hydrochloric Acid SCHEMBL2365586 0.81 HIF1A (0.52) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
Hydrochloric Acid SCHEMBL2363733 0.81 CYP3A4 (0.56) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
SCHEMBL2819013 0.80 MEN1 (0.78) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
SCHEMBL485227 0.80 CYP3A4 (0.71) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
SCHEMBL485459 0.79 CYP3A4 (0.77) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
SCHEMBL485435 0.78 HIF1A (0.67) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9
SCHEMBL484947 0.78 CYP3A4 (0.41) CYP3A4CYP2C19HIF1AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411381-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-02-01 EP disclosed
WO-2010108651-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2010-09-30 WO disclosed