SCHEMBL485898

SCHEMBL485898

CCNc1nc(-c2ccc(NC(=O)NCc3cncc(F)c3)c(F)c2)ccc1C(=O)NCCN1CCCCC1.CCNc1nc(-c2ccc(NC(=O)NCc3cncc(N)c3)c(F)c2)ccc1C(=O)NCCN1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.39
MAP4K4 O95819 1/20 0.38
TLR7 Q9NYK1 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PDE4B Q07343 3/20 0.37
ADORA2A P29274 2/20 0.37
ADORA2B P29275 2/20 0.37
ADORA1 P30542 2/20 0.37
PDPK1 O15530 1/20 0.36
CHRNA7 P36544 1/20 0.36
KCNH2 Q12809 1/20 0.36
EPHX2 P34913 1/20 0.36
SCN9A Q15858 3/20 0.35
IKBKB O14920 1/20 0.35
TGFBR1 P36897 1/20 0.35
TGFBR2 P37173 1/20 0.35
WNT1 P04628 1/20 0.35
CLK2 P49760 1/20 0.35
CLK3 P49761 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL486392 0.97 MEN1 (0.39) NAMPTMAP4K4MEN1KMT2APDE4B
SCHEMBL486297 0.96 NAMPT (0.41) NAMPTMAP4K4TLR7MEN1KMT2A
SCHEMBL485906 0.90 MEN1 (0.40) NAMPTMEN1KMT2APDE4BADORA2A
SCHEMBL486210 0.87 NAMPT (0.51) NAMPTMEN1KMT2APDE4BADORA2A
SCHEMBL3048503 0.87 NAMPT (0.50) NAMPTKCNH2EPHX2SCN9A
SCHEMBL3044891 0.87 NAMPT (0.48) NAMPTCHRNA7KCNH2EPHX2
SCHEMBL486031 0.87 MAP4K4 (0.40) MAP4K4TLR7MEN1KMT2ACHRNA7
SCHEMBL485903 0.87 PIK3CA (0.41) NAMPTMAP4K4MEN1KMT2APDPK1
SCHEMBL485908 0.87 PIK3CA (0.41) NAMPTMAP4K4MEN1KMT2APDPK1
SCHEMBL485853 0.86 PIK3CA (0.41) NAMPTMAP4K4MEN1KMT2APDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411368-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF AS ANTICANCER DRUGS SANOFI (FR) 2012-02-01 EP claimed
WO-2010109122-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF AS ANTICANCER DRUGS SANOFI-AVENTIS (FR) 2010-09-30 WO claimed