SCHEMBL4861268

SCHEMBL4861268

CC1N(c2nc(-c3ccncn3)cc(=O)n2C)CCOC1(C)C.C[C@@H]1[C@@H](C)OCCN1c1nc(-c2ccncc2F)cc(=O)n1C

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.49
CYP2D6 P10635 9/20 0.49
CYP1A2 P05177 7/20 0.49
CSNK1A1 P48729 1/20 0.48
GSK3A P49840 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL697776 0.87 GSK3B (0.56) GSK3BCYP2D6CYP1A2
SCHEMBL697777 0.87 GSK3B (0.56) GSK3BCYP2D6CYP1A2
SCHEMBL697691 0.86 GSK3B (0.62) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL8234203 0.86 GSK3B (0.62) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL8234769 0.86 GSK3B (0.62) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL698152 0.86 GSK3B (0.62) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL696630 0.86 GSK3B (0.62) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL696629 0.86 GSK3B (0.62) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL697569 0.85 GSK3B (0.62) GSK3BCYP2D6CYP1A2
SCHEMBL697684 0.85 GSK3B (0.62) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001863-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS Mitsubishi Tanabe Pharma Corporation (JP) 2008-12-17 EP disclosed
WO-2007119463-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-10-25 WO disclosed