SCHEMBL4863244

SCHEMBL4863244

COc1cc(C)c(C(=O)c2ccccc2NC(=O)c2ccc(-c3cc(-c4nnc(C)o4)ccc3C)cc2)cc1OC

nearest known ligand 0.78

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 17/20 0.78
LCK P06239 1/20 0.55
MAPK11 Q15759 2/20 0.54
ABCG2 Q9UNQ0 1/20 0.48
HTR1D P28221 1/20 0.47
CHEK1 O14757 1/20 0.45
PIM1 P11309 1/20 0.45
MAPK8 P45983 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
MAP2K1 Q02750 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4864546 0.79 MAPK14 (0.78) MAPK14LCKMAPK11HTR1DMAP2K1
SCHEMBL4855098 0.78 MAPK14 (0.77) MAPK14LCKMAPK11MAP2K1
SCHEMBL4856439 0.77 MAPK14 (1.00) MAPK14LCKMAPK11ABCG2HTR1D
SCHEMBL4856455 0.76 MAPK14 (0.74) MAPK14LCKMAPK11HTR1DMAP2K1
SCHEMBL4862307 0.76 MAPK14 (0.72) MAPK14LCKMAPK11
SCHEMBL4862266 0.76 MAPK14 (0.68) MAPK14LCKMAPK11ABCG2
SCHEMBL4861254 0.74 MAPK14 (0.67) MAPK14LCKMAPK11MAP2K1
SCHEMBL4865916 0.74 MAPK14 (0.67) MAPK14LCKMAPK11MAP2K1
SCHEMBL6605403 0.74 MAPK14 (0.67) MAPK14LCKMAPK11
SCHEMBL4862344 0.74 MAPK14 (0.69) MAPK14LCKMAPK11HTR1DMAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7384963-B2 2′-Methyl-5-(1,3,4-oxadiazol-2-yl)1, 1′-biphenyl-4-carboxaide derivatives and their use as p38 kinase GLAXO GROUP LIMITED (GB) 2008-06-10 US disclosed
US-20040266839-A1 2'-Methyl-5-(1,3,4-oxadiazol-2-yl)1,1'-biphenyl-4-carboxaide derivatives and their use as p38 kinase inhibitors GLAXO GROUP LIMITED (GB) 2004-12-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040266839-A1 2'-Methyl-5-(1,3,4-oxadiazol-2-yl)1,1'-biphenyl-4-carboxaide derivatives and their use as p38 kinase inhibitors MAPK1, MAPK3, MAPK6 MAPK14 11/4885LCK 61/4885MAPK11 17/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.