SCHEMBL4870146

SCHEMBL4870146

CC[C@@H]1C(=O)N(CC(F)(F)F)c2ccc(F)cc2N1C(=O)c1ccc(O)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.33
POLB P06746 1/20 0.33
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
PDK1 Q15118 3/20 0.32
PDK2 Q15119 3/20 0.32
PDK3 Q15120 3/20 0.32
PDK4 Q16654 3/20 0.32
HSP90AA1 P07900 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4867992 0.89 KMT2A (0.43) KMT2AMEN1POLBNR3C1PGR
SCHEMBL4862078 0.89 SMN1; SMN2 (0.39) KMT2AMEN1POLBNPC1RAB9A
SCHEMBL4869034 0.87 KMT2A (0.42) KMT2AMEN1POLBNR3C1PGR
SCHEMBL4861967 0.85 KMT2A (0.41) KMT2AMEN1POLBNR3C1PGR
SCHEMBL4867620 0.85 KMT2A (0.41) KMT2AMEN1POLB
SCHEMBL4867500 0.85 KMT2A (0.43) KMT2AMEN1POLBNR3C1PGR
SCHEMBL4867563 0.84 BRD4 (0.39) KMT2AMEN1NR3C1PGRNR3C2
SCHEMBL4869782 0.84 BRD4 (0.39) KMT2AMEN1NR3C1PGRNR3C2
SCHEMBL4865526 0.81 KMT2A (0.40) KMT2AMEN1NR3C1PGRNR3C2
SCHEMBL4864131 0.81 KMT2A (0.36) KMT2AMEN1NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7351709-B2 Estrogen receptor ligands WYETH (US) 2008-04-01 US claimed
US-20060019961-A1 Estrogen receptor ligands WYETH 2006-01-26 US claimed
US-7351709-B2 Estrogen receptor ligands WYETH (US) 2008-04-01 US disclosed
US-20060019961-A1 Estrogen receptor ligands WYETH 2006-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060019961-A1 Estrogen receptor ligands GPER1, ESR2, ESR1 KMT2A 2436/4885MEN1 4543/4885POLB 4581/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.