SCHEMBL4871197

SCHEMBL4871197

CS(=O)(=O)c1nc(C(F)(F)F)ccc1Cn1nc2c(-c3ccncc3)c(Cl)ccn2c1=O

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 19/20 0.44
CYP2C9 P11712 6/20 0.44
CYP2C19 P33261 6/20 0.44
CYP3A4 P08684 5/20 0.44
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4491848 0.87 CNR1 (0.57) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4479631 0.78 CNR1 (0.64) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4481857 0.77 CNR1 (0.64) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4491826 0.76 CNR1 (0.53) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4488160 0.75 CNR1 (0.54) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4476928 0.75 CNR1 (0.52) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4486448 0.75 CNR1 (0.53) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4478487 0.75 CNR1 (0.52) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4478611 0.75 CNR1 (0.51) CNR1CYP2C9CYP2C19CYP3A4
SCHEMBL4484312 0.75 CNR1 (0.55) CNR1CYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891068-A1 TRIAZOLOPYRIDINE DERIVATIVES AS CANNABINOID RECEPTOR 1 ANTAGONISTS Bristol-Myers Squibb Company (US) 2008-02-27 EP disclosed
WO-2006138695-A1 TRIAZOLOPYRIDINE DERIVATIVES AS CANNABINOID RECEPTOR 1 ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-12-28 WO disclosed