SCHEMBL4875601

SCHEMBL4875601

CS(=O)(=O)NCc1ccc(-c2ccccc2C(=O)NCCc2ccccc2)c(Cl)c1Cl

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
KCNA5 P22460 2/20 0.48
PTGS2 P35354 1/20 0.46
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 4/20 0.43
RCE1 Q9Y256 1/20 0.43
HPGD P15428 2/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
HSD17B10 Q99714 1/20 0.43
POLB P06746 2/20 0.42
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
PKM P14618 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4878462 0.90 KCNK3 (0.53) NPC1RAB9ALMNAKDM4EALDH1A1
SCHEMBL2208057 0.75 KCNA5 (0.72) NPC1RAB9AKCNA5MAPTALDH1A1
SCHEMBL4626781 0.73 HTT (0.68) NPC1RAB9AKCNA5MAPTLMNA
SCHEMBL2210182 0.72 KCNA5 (0.65) NPC1RAB9AKCNA5MAPTLMNA
SCHEMBL2210786 0.71 KCNA5 (0.67) NPC1RAB9AKCNA5MAPTLMNA
SCHEMBL2206886 0.70 KCNA5 (0.60) NPC1RAB9AKCNA5MAPTLMNA
SCHEMBL2205271 0.69 KCNA5 (0.59) KCNA5
SCHEMBL2210421 0.69 KCNA5 (0.60) NPC1RAB9AKCNA5MAPTHTT
SCHEMBL6356707 0.69 NPC1 (1.00) NPC1RAB9APTGS2MAPTLMNA
SCHEMBL12434478 0.67 KCNA5 (0.73) NPC1RAB9AKCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP disclosed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed