SCHEMBL4878459

SCHEMBL4878459

COc1ccc2nccc(C(O)CC3CCC(NC(=O)OC(C)(C)C)CC3)c2n1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.59
SLC2A1 P11166 4/20 0.46
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2543049 0.86 KCNH2 (0.44) KCNH2SLC2A1JAK2JAK1
SCHEMBL2543045 0.86 KCNH2 (0.44) KCNH2SLC2A1JAK2JAK1
SCHEMBL5726714 0.86 SLC2A1 (0.61) KCNH2SLC2A1
SCHEMBL16650256 0.85 KCNH2 (0.43) KCNH2SLC2A1JAK2JAK1
SCHEMBL3597040 0.85 KCNH2 (0.43) KCNH2SLC2A1JAK2JAK1
SCHEMBL16650254 0.85 KCNH2 (0.43) KCNH2SLC2A1JAK2JAK1
SCHEMBL16650253 0.85 KCNH2 (0.43) KCNH2SLC2A1JAK2JAK1
SCHEMBL2539625 0.84 KCNH2 (0.42) KCNH2SLC2A1JAK2JAK1
SCHEMBL2537316 0.84 KCNH2 (0.42) KCNH2SLC2A1JAK2JAK1
SCHEMBL2539623 0.84 KCNH2 (0.42) KCNH2SLC2A1JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987040-A1 ETHANOL OR 1,2-ETHANEDIOL CYCLOHEXYL ANTIBIOTIC DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2008-11-05 EP disclosed
WO-2007093963-A1 ETHANOL OR 1,2-ETHANEDIOL CYCLOHEXYL ANTIBIOTIC DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2007-08-23 WO disclosed