SCHEMBL4879216

SCHEMBL4879216

Cc1cn(-c2cc(C(=O)Nc3ccc(C)c(Nc4ccnc(-c5cncnc5)n4)c3)cc(C(F)(F)F)c2)cn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 9/20 0.61
CSF1R P07333 2/20 0.60
KDM4E B2RXH2 1/20 0.60
POLB P06746 1/20 0.60
RECQL P46063 1/20 0.60
BCR P11274 5/20 0.59
BRAF P15056 4/20 0.59
HCK P08631 4/20 0.59
RAF1 P04049 3/20 0.59
LCK P06239 3/20 0.59
LYN P07948 3/20 0.59
SRC P12931 3/20 0.59
ADORA3 P0DMS8 2/20 0.59
LDLR P01130 2/20 0.59
PDGFRB P09619 2/20 0.59
KIT P10721 2/20 0.59
PCSK9 Q8NBP7 2/20 0.59
EPHB2 P29323 2/20 0.59
FYN P06241 2/20 0.59
YES1 P07947 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630979 0.83 BRAF (0.68) ABL1CSF1RPOLBBRAFRAF1
SCHEMBL5222415 0.83 ABL1 (0.84) ABL1CSF1RBCRBRAFHCK
SCHEMBL15381989 0.79 CSF1R (0.71) ABL1CSF1RKDM4EPOLBRECQL
SCHEMBL22025121 0.78 ABL1 (0.63) ABL1CSF1RKDM4EPOLBRECQL
SCHEMBL6451143 0.78 KDM4E (0.64) ABL1CSF1RKDM4EPOLBRECQL
SCHEMBL27708222 0.78 PIKFYVE (0.55) ABL1CSF1RBCRBRAFPDGFRB
SCHEMBL2465750 0.78 LCK (0.70) CSF1RKDM4EPOLBRECQLHCK
SCHEMBL15556278 0.77 EPHB2 (0.82) ABL1CSF1RKDM4EPOLBRECQL
SCHEMBL21612152 0.76 CSF1R (0.71) ABL1CSF1RKDM4EPOLBRECQL
SCHEMBL4252904 0.76 CSF1R (0.68) ABL1CSF1RKDM4EPOLBRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080146570-A1 Chemical Compounds ASTRAZENECA AB (SE) 2008-06-19 US claimed
US-20080146570-A1 Chemical Compounds ASTRAZENECA AB (SE) 2008-06-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080146570-A1 Chemical Compounds BRAF, RAF1, NRAS ABL1 20/4885CSF1R 1706/4885KDM4E 2971/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.