Dilazep

Dilazep

SCHEMBL48830

COc1cc(C(=O)OCCCN2CCCN(CCCOC(=O)c3cc(OC)c(OC)c(OC)c3)CC2)cc(OC)c1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 10/20 1.00
MEN1 O00255 5/20 1.00
KMT2A Q03164 5/20 1.00
SMN1; SMN2 Q16637 4/20 1.00
CYP2D6 P10635 4/20 1.00
CYP3A4 P08684 3/20 1.00
LMNA P02545 2/20 1.00
SCN1A P35498 2/20 1.00
SCN2A Q99250 2/20 1.00
SCN3A Q9NY46 2/20 1.00
THPO P40225 2/20 1.00
MTOR P42345 2/20 1.00
ABCC4 O15439 1/20 1.00
CYP2C9 P11712 1/20 1.00
TSHR P16473 1/20 1.00
CHRM3 P20309 1/20 1.00
HTR2A P28223 1/20 1.00
MAPK1 P28482 1/20 1.00
SLC6A4 P31645 1/20 1.00
CYP2C19 P33261 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dilazep SCHEMBL2597896 1.00 SLC29A1 (1.00) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
Dilazep SCHEMBL220842 0.99 SMN1; SMN2 (1.00) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
Dilazep SCHEMBL349239 0.99 SMN1; SMN2 (1.00) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
Dilazep SCHEMBL9934077 0.97 SMN1; SMN2 (0.98) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
Dilazep SCHEMBL15532226 0.97 SLC29A1 (0.95) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
SCHEMBL27319577 0.93 SLC29A1 (0.87) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
SCHEMBL2459734 0.91 SLC29A1 (0.83) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
SCHEMBL27319054 0.91 SLC29A1 (0.83) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
SCHEMBL8686213 0.88 SLC29A1 (0.79) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6
Dilazep SCHEMBL11130839 0.87 SLC29A1 (0.77) SLC29A1MEN1KMT2ASMN1; SMN2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4688 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12550885-B2 Red blood cell storage solutions, solution additives, and methods for improving the storage of red blood cells UNIVERSITY OF CINCINNATI (US) 2026-02-17 US claimed
WO-2025262072-A2 NEURONAL DRUG SCREENING METHOD AND NEW APPLICATIONS FOR DILAZEP AND PENBUTOLOL MIĘDZYNARODOWY INSTYTUT BIOLOGII MOLEKULARNEJ I KOMÓRKOWEJ (PL) 2025-12-26 WO claimed
EP-4658278-A1 SELECTIVE FIASMA TREATMENT Valo Health, Inc. (US) 2025-12-10 EP claimed
US-12480096-B2 Clinical gene signature-based human cell culture model and uses thereof UNIVERSITE DE STRASBOURG (FR) 2025-11-25 US claimed
WO-2025202864-A1 ENT1 INHIBITORS IN COMBINATION WITH ONCOLYTIC VIRUSES AND THEIR USE IN THE TREATMENT OF CANCER iTeos Belgium SA (BE) 2025-10-02 WO claimed
WO-2025074343-A2 PRODRUGS OF HUMAN DIHYDROOROTATE DEHYDROGENASE (hDHODH) INHIBITORS DRUG DISCOVERY AND CLINIC S.R.L. (IT) 2025-04-10 WO claimed
WO-2024163699-A1 SELECTIVE FIASMA TREATMENT VALO HEALTH, INC. (US) 2024-08-08 WO claimed
EP-4387735-A2 ANTIVIRAL DRUGS TARGETING THE N-TERMINAL DOMAIN (NTD) OF THE CORONAVIRUS SPIKE RECEPTOR BINDING DOMAIN (RBD) SOUTHWEST RESEARCH INSTITUTE (US) 2024-06-26 EP claimed
US-20230321008-A1 INHIBITORS OF ACID SPHINGOMYELINASE FOR PREVENTING AND TREATING THE COVID-19 DISEASE ASSISTANCE PUBLIQUE - HOPITAUX DE PARIS (FR) 2023-10-12 US claimed
WO-2023183932-A2 MONOBODIES BINDING TO INTERCELLULAR ADHESION MOLECULE 2 (ICAM-2) NEW YORK UNIVERSITY (US) 2023-09-28 WO claimed
WO-1989010122-A1 COMPOSITIONS AND METHODS FOR TREATING CUTANEOUS HYPERPROLIFERATIVE DISORDERS YALE UNIVERSITY (US) 1989-11-02 WO claimed
US-4873228-A 2-oxo-4-carboxy-pyrimidines and their use as anti-malaria and anti-cancer agents THE UNIVERSITY OF MELBOURNE (AU) 1989-10-10 US claimed
EP-0170361-B1 ANTIATHEROSCLEROTIC AGENTS KOWA COMPANY, LTD. (JP) 1989-08-02 EP claimed
US-4751298-A Production of 1-(3-hydroxy-propyl)-1,4-diazepane and 1,4-bis(3,4,5-trimethoxy-benzoyloxy)-propyl-diazepane derivatives thereof DEGUSSA AKTIENGESELLSCHAFT (DE) 1988-06-14 US claimed
US-4751224-A FORSKOLIN DERIVATIVES; ANTIAGGLOMERANTS BROWN UNIVERSITY RESEARCH FOUNDATION (US) 1988-06-14 US claimed
EP-0235931-A1 Antiviral combination THE WELLCOME FOUNDATION LIMITED (GB) 1987-09-09 EP claimed
EP-0217580-A2 Therapeutic nucleosides THE WELLCOME FOUNDATION LIMITED (GB) 1987-04-08 EP claimed
EP-0170361-A1 Antiatherosclerotic agents KOWA COMPANY, LTD. (JP) 1986-02-05 EP claimed
EP-0167567-A1 TREATMENT OF METASTASIS BROWN UNIVERSITY RESEARCH FOUNDATION (US) 1986-01-15 EP claimed
WO-1985002616-A1 TREATMENT OF METASTASIS BROWN UNIVERSITY RESEARCH FOUNDATION (US) 1985-06-20 WO claimed