SCHEMBL4884233

SCHEMBL4884233

Cc1ccc(N)cc1-n1cnc2ccc(Br)cc2c1=O

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 3/20 0.45
MAPK14 Q16539 10/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MCL1 Q07820 1/20 0.41
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4829534 0.83 POLB (0.51) MEN1KMT2A
SCHEMBL4886749 0.82 MAPK14 (0.52) MAPK14MCL1
SCHEMBL1140575 0.79 MAPK14 (0.52) MAPK14MCL1
SCHEMBL4827748 0.78 MAPK14 (0.69) MAPK14
SCHEMBL4827243 0.75 MAPK14 (0.65) MAPK14
SCHEMBL3656842 0.72 MEN1 (0.68) HCAR1MEN1KMT2AMCL1ATM
SCHEMBL4887021 0.71 SCD (0.62) MAPK14
SCHEMBL4879776 0.71 MAPK14 (0.49) MAPK14
SCHEMBL16204799 0.70 MEN1 (0.55) HCAR1MEN1KMT2AMCL1
SCHEMBL3751890 0.70 CHEK1 (0.51) MEN1KMT2AMCL1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080275022-A1 Substituted Quinazolones as Anti-Cancer Agents ASTRAZENECA AB (SE) 2008-11-06 US disclosed
CN-101001845-A Substituted quinazolones as anti-cancer agents. ASTRAZENECA AB (SE) 2007-07-18 CN disclosed
EP-1761506-A1 SUBSTITUTED QUINAZOLONES AS ANTI-CANCER AGENTS AstraZeneca AB (SE) 2007-03-14 EP disclosed
WO-2005123696-A1 SUBSTITUTED QUINAZOLONES AS ANTI-CANCER AGENTS ASTRAZENECA AB (SE) 2005-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080275022-A1 Substituted Quinazolones as Anti-Cancer Agents BRAF, NRAS, RAF1 HCAR1 4034/4885MAPK14 153/4885MEN1 872/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.