SCHEMBL4891653

SCHEMBL4891653

Cc1ccc(NC(=O)c2cccnc2)cc1Nc1nccc(-c2ccc(-n3ccnc3)cc2)n1

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 13/20 0.70
ABL1 P00519 11/20 0.70
BCR P11274 7/20 0.70
PDGFRB P09619 6/20 0.70
EGFR P00533 2/20 0.70
PRKCA P17252 1/20 0.70
KIT P10721 5/20 0.62
LCK P06239 1/20 0.60
LYN P07948 1/20 0.60
FLT3 P36888 1/20 0.60
DDR2 Q16832 1/20 0.60
KDR P35968 1/20 0.58
ABL2 P42684 1/20 0.58
JAK3 P52333 1/20 0.58
BTK Q06187 1/20 0.58
ITK Q08881 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4901347 0.89 PDGFRA (0.69) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4897554 0.89 ABL1 (0.72) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4903594 0.89 KIT (0.59) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4900996 0.88 PDGFRA (0.70) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL2004455 0.87 PDGFRA (0.91) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL17263675 0.85 ABL1 (0.81) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4902240 0.85 ABL1 (0.71) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4899621 0.85 PDGFRA (0.57) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4903220 0.85 PDGFRA (0.55) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL3533748 0.84 ABL1 (0.70) PDGFRAABL1BCRPDGFRBEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080187575-A1 Pyrimidine Derivatives VICHEM CHEMIE KFT (HU) 2008-08-07 US claimed
US-20080187575-A1 Pyrimidine Derivatives VICHEM CHEMIE KFT (HU) 2008-08-07 US disclosed
EP-1786781-A2 PYRIMIDINE DERIVATIVES GPC Biotech AG (DE) 2007-05-23 EP disclosed
WO-2006021458-A2 PYRIMIDINE DERIVATIVES GPC BIOTECH AG (DE) 2006-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080187575-A1 Pyrimidine Derivatives TYMP, TDP1, PNP PDGFRA 373/4885ABL1 2843/4885BCR 2315/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.