Zenarestat

Zenarestat

SCHEMBL48959

O=C(O)Cn1c(=O)n(Cc2ccc(Br)cc2F)c(=O)c2ccc(Cl)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 8/20 1.00
AKR1A1 P14550 1/20 1.00
HDAC6 Q9UBN7 3/20 0.48
AKR1B10 O60218 2/20 0.46
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HDAC1 Q13547 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
MAPK8 P45983 1/20 0.42
MAPK9 P45984 1/20 0.42
OPRM1 P35372 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90B1 P14625 1/20 0.41
TRAP1 Q12931 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Zenarestat SCHEMBL29688249 1.00 AKR1B1 (1.00) AKR1B1AKR1A1HDAC6AKR1B10MEN1
Zenarestat SCHEMBL30583313 1.00 AKR1B1 (1.00) AKR1B1AKR1A1HDAC6AKR1B10MEN1
SCHEMBL10487878 0.92 AKR1B1 (0.86) AKR1B1AKR1A1HDAC6AKR1B10MEN1
SCHEMBL10488007 0.92 AKR1B1 (0.85) AKR1B1AKR1A1HDAC6AKR1B10MEN1
Zenarestat SCHEMBL10487895 0.90 AKR1B1 (0.81) AKR1B1AKR1A1HDAC6AKR1B10MEN1
SCHEMBL9319101 0.89 AKR1B1 (0.81) AKR1B1AKR1A1HDAC6AKR1B10MEN1
SCHEMBL10487834 0.88 AKR1B1 (0.79) AKR1B1AKR1A1AKR1B10MEN1CYP1A2
SCHEMBL10487869 0.88 AKR1B1 (0.78) AKR1B1AKR1A1HDAC6AKR1B10MEN1
SCHEMBL10487836 0.88 AKR1B1 (0.78) AKR1B1AKR1A1HDAC6AKR1B10MEN1
SCHEMBL9056716 0.88 AKR1B1 (0.78) AKR1B1AKR1A1HDAC6AKR1B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2944 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240374693-A1 TREATMENT AND DETECTION OF INHERITED NEUROPATHIES AND ASSOCIATED DISORDERS UNIVERSITY OF ROCHESTER 2024-11-14 US claimed
US-12083168-B2 Treatment and detection of inherited neuropathies and associated disorders UNIVERSITY OF MIAMI (US) 2024-09-10 US claimed
WO-2024053761-A1 COMPOSITION FOR PROMOTING MYOBLAST PROLIFERATION AND DIFFERENTIATION CONTAINING ALDOSE REDUCTASE INHIBITOR 애니머스큐어 주식회사 2024-03-14 WO claimed
US-20240003908-A1 POLYOL BIOMARKERS FOR CONGENITAL DISORDERS OF GLYCOSYLATION MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH 2024-01-04 US claimed
US-20230293642-A9 TREATMENT AND DETECTION OF INHERITED NEUROPATHIES AND ASSOCIATED DISORDERS UNIVERSITY OF ROCHESTER 2023-09-21 US claimed
EP-4244243-A1 POLYOL BIOMARKERS FOR CONGENITAL DISORDERS OF GLYCOSYLATION Mayo Foundation for Medical Education and Research (US) 2023-09-20 EP claimed
US-20220249624-A1 TREATMENT AND DETECTION OF INHERITED NEUROPATHIES AND ASSOCIATED DISORDERS UNIV MIAMI (US) 2022-08-11 US claimed
WO-2022103815-A1 POLYOL BIOMARKERS FOR CONGENITAL DISORDERS OF GLYCOSYLATION MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2022-05-19 WO claimed
US-20220125890-A1 TREATMENT AND DETECTION OF INHERITED NEUROPATHIES AND ASSOCIATED DISORDERS UNIVERSITY OF ROCHESTER 2022-04-28 US claimed
US-20220125766-A1 METHODS FOR TREATING CONGENITAL DISORDERS OF GLYCOSYLATION MAGGIES PEARL LLC (US) 2022-04-28 US claimed
EP-1097707-A1 Treatment of female sexual dysfunction Pfizer Limited (GB) 2001-05-09 EP claimed
US-6218409-B1 ADMINISTERING INSULIN SENSITIVITY ENHANCER IN COMBINATION WITH AN ALDOSE REDUCTASE INHIBITOR FOR REDUCING SIDE EFFECTS OF DIABETIC DRUGS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-17 US claimed
US-6156773-A Pharmaceutical composition TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-05 US claimed
WO-2000045818-A1 USE OF 3-HYDROXY-3-METHYLGLUTARYL COENZYM A REDUCTASE INHIBITORS FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF DIABETIC NEUROPATHY ASTRAZENECA AB (SE) 2000-08-10 WO claimed
CN-1261804-A Pharmaceutical compositions comprising an aldose reductase inhibitor and an ACE inhibitor ZENECA LTD (GB) 2000-08-02 CN claimed
WO-2000037066-A2 A METHOD FOR THE PROPHYLACTIC TREATMENT OF CATARACTS JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2000-06-29 WO claimed
EP-0991424-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING AN ALDOSE REDUCTASE INHIBITOR AND AN ACE INHIBITOR ZENECA LIMITED (GB) 2000-04-12 EP claimed
WO-1999002189-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING AN ALDOSE REDUCTASE INHIBITOR AND AN ACE INHIBITOR ZENECA LIMITED (GB) 1999-01-21 WO claimed
US-4734419-A Quinazoline derivatives, compositions thereof and their use in treating diabetic complications FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-03-29 US claimed
EP-0218999-A2 New quinazoline derivatives, process for their production and pharmaceutical compositions comprising them FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-04-22 EP claimed