SCHEMBL4899602

SCHEMBL4899602

Cc1ccc(NC(=O)c2ccccc2)cc1Nc1nccc(-c2ccncc2)n1

nearest known ligand 0.82

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 13/20 0.82
ABL1 P00519 11/20 0.82
BCR P11274 7/20 0.82
PDGFRB P09619 6/20 0.82
PRKCA P17252 2/20 0.82
EGFR P00533 1/20 0.82
KIT P10721 5/20 0.66
KDR P35968 1/20 0.62
ABL2 P42684 1/20 0.62
JAK2 O60674 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4897274 0.92 PDGFRA (0.80) PDGFRAABL1BCRPDGFRBPRKCA
SCHEMBL4900883 0.90 PDGFRA (0.81) PDGFRAABL1BCRPDGFRBPRKCA
SCHEMBL29498750 0.90 PDGFRA (1.00) PDGFRAABL1BCRPDGFRBPRKCA
SCHEMBL9782 0.90 PDGFRA (1.00) PDGFRAABL1BCRPDGFRBPRKCA
Methane SCHEMBL5972158 0.89 PDGFRA (0.98) PDGFRAABL1BCRPDGFRBPRKCA
SCHEMBL4905638 0.88 PDGFRA (0.67) PDGFRAABL1BCRPDGFRBPRKCA
SCHEMBL4903357 0.88 PDGFRA (0.66) PDGFRAABL1BCRPDGFRBPRKCA
SCHEMBL5187795 0.86 PDGFRA (0.73) PDGFRAABL1BCRPDGFRBPRKCA
SCHEMBL4899291 0.86 ABL1 (0.62) PDGFRAABL1BCRPDGFRBPRKCA
SCHEMBL5189023 0.85 PDGFRA (0.85) PDGFRAABL1BCRPDGFRBPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080187575-A1 Pyrimidine Derivatives VICHEM CHEMIE KFT (HU) 2008-08-07 US claimed
EP-1786781-A2 PYRIMIDINE DERIVATIVES GPC Biotech AG (DE) 2007-05-23 EP claimed
WO-2006021458-A2 PYRIMIDINE DERIVATIVES GPC BIOTECH AG (DE) 2006-03-02 WO claimed
US-20080187575-A1 Pyrimidine Derivatives VICHEM CHEMIE KFT (HU) 2008-08-07 US disclosed
EP-1786781-A2 PYRIMIDINE DERIVATIVES GPC Biotech AG (DE) 2007-05-23 EP disclosed
WO-2006021458-A2 PYRIMIDINE DERIVATIVES GPC BIOTECH AG (DE) 2006-03-02 WO disclosed
EP-1395261-A2 PYRIDYLPYRIMIDINE DERIVATIVES AS EFFECTIVE COMPOUNDS AGAINST PRION DISEASES Axxima Pharmaceuticals Aktiengesellschaft (DE) 2004-03-10 EP disclosed
WO-2002093164-A2 PYRIDYLPYRIMIDINE DERIVATIVES AS EFFECTIVE COMPOUNDS AGAINST PRION DISEASES AXXIMA PHARMACEUTICALS AG (DE) 2002-11-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080187575-A1 Pyrimidine Derivatives TYMP, TDP1, PNP PDGFRA 373/4885ABL1 2843/4885BCR 2315/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.